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Naltrexone is a medication that blocks the effects of drugs known as opioids (a class that includes morphine, heroin or codeine). It competes with these drugs for opioid receptors in the brain. ... Second, naltrexone helps patients remain abstinent.
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In terms of dosing, 50mg of naltrexone have the ability to block the effects of opioids for about 24 hours. Clinical studies suggest that doubling the dose will block opioid effects for 48 hours, while 150mg of naltrexone can provide blockage for approximately 72 hours.
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